S. No | Inhibitor IUPAC Name | Ki values (mM) |
---|---|---|
Inh-1 | 2-oxobutanoate | 0.83 |
Inh-2 | 2-oxoheptanedioate | 0.17 |
Inh-3 | 2-oxopentanoate | 0.7 |
Inh-4 | 3-bromo-2-oxopropanoate | 1.6 |
Inh-5 | 3-fluoro-2-oxopropanoate | 0.22 |
Inh-6 | 2,4-dioxopentanoic acid | 0.005 |
Inh-7 | (2R)-2-amino-3-(2-aminoethylsulfanyl)propanoic acid | 2.4 |
Inh-8 | (2S)-2-aminocyclopentan-1-one | 12 |
Inh-9 | (2R)-2-azaniumyl-4-hydroxy-4-oxobutanoate | 0.09 |
Inh-10 | 4-oxo-1H-pyridine-2,6-dicarboxylic acid | 22 |
Inh-11 | 2,6-dioxoheptanedioic acid | 0.156 |
Inh-12 | Dimethyl 4-oxo-1H-pyridine-2,6-dicarboxylate | 6.9 |
Inh-13 | Pyridine-2,6-dicarbonitrile | 0.35 |
Inh-14 | Pyridine-2,6-dicarboxylate | 11 |
Inh-15 | Oxaldehydate | 0.028 |
Inh-16 | (3R)-3-aminooxolan-2-one | 8 |
Inh-17 | Benzene-1,3-dicarboxylic acid | 15 |
Inh-18 | (2S)-2-amino-4-oxobutanoic acid | 0.27 |
Inh-19 | 1-oxidopyridin-1-ium-2,6-dicarboxylic acid | 0.06 |
Inh-20 | (2S)-2-azaniumyl-3 sulfinopropanoate | 6.1 |
Inh-21 | (2S)-2-azaniumyl-5-hydroxy-5-oxopentanoate | 9 |
Inh-22 | 4-oxobutanoic acid | 0.3 |
Inh-23 | (1R)-cyclohex-3-ene-1,3-dicarboxylic acid | 15 |